Preparation of 18F-labeled muscarinic agonist with M2 selectivity

J Med Chem. 1995 Jan 6;38(1):5-8. doi: 10.1021/jm00001a002.
No abstract available

MeSH terms

  • Animals
  • Brain / metabolism
  • Fluorine Compounds / chemical synthesis*
  • Fluorine Compounds / pharmacology*
  • Fluorine Radioisotopes
  • Isotope Labeling
  • Kinetics
  • Muscarinic Agonists* / chemical synthesis*
  • Muscarinic Agonists* / pharmacology*
  • Pyridines / chemical synthesis*
  • Pyridines / pharmacology*
  • Rats
  • Rats, Sprague-Dawley
  • Receptors, Muscarinic / classification
  • Receptors, Muscarinic / metabolism
  • Sensitivity and Specificity
  • Thiadiazoles / chemical synthesis*
  • Thiadiazoles / pharmacology*
  • Tissue Distribution

Substances

  • Fluorine Compounds
  • Fluorine Radioisotopes
  • Muscarinic Agonists
  • Pyridines
  • Receptors, Muscarinic
  • Thiadiazoles